Publication

業績

国嶋崇隆 教授

  1. Effects of the (Trialkyl)ammonium Structures in (Ammonio)amidyl Groups on π-Electron Donating Ability and Thermal Stability: Experimental and Computational Study
    Hikaru Fujita, Takanari Arai, Hiroki Muraya, Yoshika Matsuyama, Munetaka KunishimaChemical and Pharmaceutical Bulletin 2025年8月29日  
  2. Development of a Triazinyluronium-Based Dehydrative Condensing Reagent with No Heteroatomic Bonds
    Gaku Mizushima, Hikaru Fujita, Munetaka KunishimaThe Journal of Organic Chemistry 2024年12月20日  
  3. Alkoxy Exchange Strategy for the Synthesis of N,N′-Dimethylated (Alkoxy)triazinediones as Solid Reagents for Acid-Catalyzed O-Alkylation
    Hikaru Fujita, Tomomi Yagitani, Munetaka KunishimaThe Journal of Organic Chemistry 2024年10月1日  
  4. Bicyclic-Ammonium-Incorporated Ylidic Nitrogen Groups for Strong π-Electron Donation in Push–Pull Benzene π-Conjugated Systems
    Hikaru Fujita, Takanari Arai, Naoto Kuchiki, Munetaka KunishimaOrganic Letters 2024年8月26日  
  5. Phototriggered Generation of Ynol Ethers and Their Rearrangement to Ketenes.
    Shunsuke Mogami, Masanobu Baba, Taniyuki Furuyama, Munetaka Kunishima, Kenji MishiroThe Journal of organic chemistry 2024年7月16日  
  6. Development of a Purely Isolable (Dimorpholino)triazine-Based Reagent for the Epoxidation of Alkenes
    Hikaru Fujita, Toshiyuki Kato, Tatsuki Betsuyaku, Munetaka KunishimaSynlett 2024年6月28日  
  7. Development of radioiodine-labeled mequitazine for evaluation of hepatic CYP2D activity
    Asuka Mizutani, Masato Kobayashi, Kodai Nishi, Ken-ichi Fujita, Kotaro Takahashi, Yuka Muranaka, Kakeru Sato, Masanori Kitamura, Chie Suzuki, Ryuichi Nishii …Frontiers in Pharmacology 15 2024年6月19日  
  8. Carbocationoids, a concept for controlling highly reactive cationic species
    Hikaru Fujita, Daichi Shimada, Jotaro Kudo, Kazuyuki Kosha, Satoshi Kakuyama, Hiromitsu Terasaki, Munetaka KunishimaCommunications Chemistry 7(1) 2024年3月13日  
  9. Drug–drug conjugates of MEK and Akt inhibitors for RAS-mutant cancers
    Hikaru Fujita, Sachiko Arai, Hiroshi Arakawa, Kana Hamamoto, Toshiyuki Kato, Tsubasa Arai, Nanaka Nitta, Kazuki Hotta, Natsuko Hosokawa, Takako Ohbayashi …Bioorganic & Medicinal Chemistry 102 117674-117674 2024年3月  
  10. Phototriggered Butenolide Formation from a Cyclobutenedione and an Acidic Nucleophile.
    Kenji Mishiro, Aiko Sesumi, Takanori Fujii, Taniyuki Furuyama, Munetaka KunishimaOrganic letters 26(1) 380-384 2024年1月12日  
  11. Epitope-Based Specific Antibody Modifications.
    Saki Horie, Kenji Mishiro, Mio Nishino, Inori Domae, Mitsuo Wakasugi, Tsukasa Matsunaga, Munetaka KunishimaBioconjugate chemistry 34(11) 2022-2033 2023年11月15日  
  12. Synthesis and characterization of tetraphenylammonium salts
    Hikaru Fujita, Ozora Sasamoto, Shiori Kobayashi, Masanori Kitamura, Munetaka KunishimaNature Communications 13(1) 2022年12月  
  13. Hydrophobic‐Substrate‐Selective Dehydrative Condensations at the Emulsion Interface under Conditions where Competitive Reactions Proceed in the Bulk Aqueous Phase
    Takuya Matsumoto, Eri Hirata, Hanlin Zhang, Kazuhito Hioki, Munetaka KunishimaAsian Journal of Organic Chemistry 2022年11月14日  
  14. Measurement of Hepatic CYP3A4 and 2D6 Activity Using Radioiodine-Labeled O-Desmethylvenlafaxine.
    Asuka Mizutani, Masato Kobayashi, Riku Aibe, Yuka Muranaka, Kodai Nishi, Masanori Kitamura, Chie Suzuki, Ryuichi Nishii, Naoto Shikano, Yasuhiro Magata …International journal of molecular sciences 23(19) 2022年9月28日  
  15. Ideal Thesis Research and Clinical Training as Pharmaceutical Practice in 6-year Pharmaceutical Education and Study System
    Munetaka KunishimaYAKUGAKU ZASSHI 142(8) 821-827 2022年8月1日  
  16. Discovery of a Novel Aminocyclopropenone Compound That Inhibits BRD4-Driven Nucleoporin NUP210 Expression and Attenuates Colorectal Cancer Growth
    Kondo, H., Mishiro, K., Iwashima, Y., Qiu, Y., Kobayashi, A., Lim, K., Domoto, T., Minamoto, T., Ogawa, K., Kunishima, M. …Cells 11(3) 317-317 2022年  
  17. Synthesis of N-Aminated Salts of Aliphatic tert-Amines, (Trialkyl)amidines, and (Pentaalkyl)guanidines by Electrophilic Amination in an Ethereal Solvent
    Fujita, H., Arai, T., Kunishima, M.Chemical and Pharmaceutical Bulletin 70(1) 85-88 2022年  
  18. Nucleophilic substitution reactions of unbranched alkyl amines using triazine reagents
    Kitamura, M., Kitaoka, Y., Fujita, H., Kunishima, M.Tetrahedron Letters 93 153692-153692 2022年  
  19. 2,4,6‐Tris( p ‐methoxybenzyloxy)‐1,3,5‐triazine (TriBOT‐PM)
    Hikaru Fujita, Munetaka KunishimaEncyclopedia of Reagents for Organic Synthesis 1-3 2021年5月17日  
  20. N-Acyltriazinedione; a Novel Acylating Reagent Synthesized from a Triazinone-Type Condensing Reagent
    Kohei Yamada, Jeongsu Lee, Mika Kota, Yukiko Karuo, Masanori Kitamura, Munetaka KunishimaChemical and Pharmaceutical Bulletin 69(5) 498-502 2021年5月1日  
  21. Efficiency Enhancement of a Photocatalytic Decarbonylation of an Aminocyclopropenone by Benzothiophene Substitution.
    Kenji Mishiro, Mitsuki Nomura, Taniyuki Furuyama, Munetaka KunishimaThe Journal of organic chemistry 86(4) 3625-3636 2021年2月19日  
  22. Conjugation of 4-(dimethylamino)pyridine to primary amines in aqueous buffer solutions using an N-hydroxysuccinimide ester reagent
    Horie, S., Fujita, H., Yamashita, R., Kunishima, M.Tetrahedron Letters 81 2021年  
  23. Development of a triazinedione-based dehydrative condensing reagent containing 4-(dimethylamino)pyridine as an acyl transfer catalyst
    Jie Liu, Hikaru Fujita, Masanori Kitamura, Daichi Shimada, Munetaka KunishimaOrganic & Biomolecular Chemistry 19(21) 4712-4719 2021年  
  24. A versatile iodo(iii)etherification of terminal ethynylsilanes using BF3–OiPr2 and alkyl benzyl ethers
    Takuya Matsumoto, Hiroshi Hagiyama, Kanetsugu Kuribayashi, Kazuhito Hioki, Hikaru Fujita, Masahito Ochiai, Munetaka KunishimaOrganic & Biomolecular Chemistry 2021年  
  25. 6-Hydroxyindole is an endogenous long-lasting OATP1B1 inhibitor elevated in renal failure patients.
    Yusuke Masuo, Ken-Ichi Fujita, Kenji Mishiro, Natsumi Seba, Tatsuya Kogi, Hidenori Okumura, Natsumi Matsumoto, Munetaka Kunishima, Yukio KatoDrug metabolism and pharmacokinetics 35(6) 555-562 2020年12月  
  26. Trizaine-based dehydrative condensation reagents bearing carbon-substituents
    Masanori Kitamura, Sayaka Komine, Kohei Yamada, Munetaka KunishimaTetrahedron 76(12) 130900-130900 2020年3月  
  27. Development of Hydrophilic Polyacrylamide Gel-Based Condensing Reagents Comprised of Chlorotriazine.
    Kohei Yamada, Shota Hirozawa, Junqing Xia, Munetaka KunishimaChemical & pharmaceutical bulletin 68(6) 534-537 2020年  
  28. Development of Triazinone-Based Condensing Reagents for Amide Formation
    Kohei Yamada, Mika Kota, Kensuke Takahashi, Hikaru Fujita, Masanori Kitamura, Munetaka KunishimaThe Journal of Organic Chemistry 84(23) 15042-15051 2019年12月6日  
  29. Preparation of Alkyl Ethers with Diallyltriazinedione-Type Alkylating Agents (ATTACKs-R) Under Acid Catalysis
    Fujita Hikaru, Yamashita Rina, Fujii Takanori, Yamada Kohei, Kitamura Masanori, Kunishima MunetakaEUROPEAN JOURNAL OF ORGANIC CHEMISTRY (27) 4436-4446 2019年7月23日  
  30. Substitution of the Dimethylamino Group in Gramines and One-Pot Cyclization to Tetrahydro-beta-carbolines Using a Triazine-Based Activating Agent
    Fujita Hikaru, Nishikawa Riho, Sasamoto Ozora, Kitamura Masanori, Kunishima MunetakaJOURNAL OF ORGANIC CHEMISTRY 84(13) 8380-8391 2019年7月5日  
  31. Substitution of the Dimethylamino Group in Gramines and One-Pot Cyclization to Tetrahydro-β-carbolines Using a Triazine-Based Activating Agent.
    Fujita H, Nishikawa R, Sasamoto O, Kitamura M, Kunishima MThe Journal of organic chemistry 84(13) 8380-8391 2019年7月5日  
  32. Phototriggered Active Alkyne Generation from Cyclopropenones with Visible Light-Responsive Photocatalysts.
    Mishiro K, Kimura T, Furuyama T, Kunishima MOrganic letters 21(11) 4101-4105 2019年6月7日  
  33. Development of a Storable Triazinone-Based Reagent for O-p-Methoxybenzylation under Mild Heating Conditions
    Fujita Hikaru, Terasaki Hiromitsu, Kakuyama Satoshi, Hioki Kazuhito, Kunishima MunetakaORGANIC LETTERS 21(9) 3093-3097 2019年5月3日  
  34. Development of a Storable Triazinone-Based Reagent for O- p-Methoxybenzylation under Mild Heating Conditions.
    Fujita H, Terasaki H, Kakuyama S, Hioki K, Kunishima MOrganic letters 21(9) 3093-3097 2019年5月3日  
  35. Phototriggered Active Alkyne Generation from Cyclopropenones with Visible Light-Responsive Photocatalysts.
    Kenji Mishiro, Takeshi Kimura, Taniyuki Furuyama, Munetaka KunishimaOrganic letters 21(11) 4101-4105 2019年5月  
  36. Triazine-Based Cationic Leaving Group: Synergistic Driving Forces for Rapid Formation of Carbocation Species
    Fujita Hikaru, Kakuyama Satoshi, Fukuyoshi Shuichi, Hayakawa Naoko, Oda Akifumi, Kunishima MunetakaJournal of Organic Chemistry 83(8) 4568-4580 2018年  
  37. Development of radioiodine labeled acetaminophen for specific, high-contrast imaging of malignant melanoma
    Zhu Wen Jing, Kobayashi Masato, Yamada Kohei, Nishi Kodai, Takahashi Kotaro, Mizutani Asuka, Nishii Ryuichi, Flores Leo G. II, Shikano Naoto, Kunishima Munetaka …Nuclear Medicine and Biology 59 16-21 2018年  
  38. An Isolable and Bench-Stable Epoxidizing Reagent Based on Triazine: Triazox
    Yamada Kohei, Igarashi Yuki, Betsuyaku Tatsuki, Kitamura Masanori, Hirata Koki, Hioki Kazuhito, Kunishima MunetakaOrganic Letters 20(7) 2015-2019 2018年  
  39. Development of Triazine-Based Benzylating Reagents Possessing t-Butyl Group on the Triazine Core: Thermally Controllable Reagents for the Initiation of Reaction
    Karuo Yukiko, Yamada Kohei, Kunishima MunetakaChemical & Pharmaceutical Bulletin 66(3) 303-308 2018年  
  40. Development of highly electron-deficient and less sterically-hindered phosphine ligands possessing 1,3,5-triazinyl groups
    Abe Kazumi, Kitamura Masanori, Fujita Hikaru, Kunishima MunetakaMolecular Catalysis 445 87-93 2018年  
  41. Cooperation of the Neutral and the Cationic Leaving Group Pathways in Acid-Catalyzed O-Benzylation of TriBOT.
    Fujita H, Hayakawa N, Kunishima MThe Journal of organic chemistry 83(17) 10684-10687 2018年  
  42. Development of triazine-based esterifying reagents containing pyridines as a nucleophilic catalyst.
    Yamada K, Liu J, Kunishima MOrganic & biomolecular chemistry 16(35) 6569-6575 2018年  
  43. Phototriggered Ketone Formation from an Aminocyclopropenone and a Carboxylic Acid.
    Mishiro K, Yushima Y, Kunishima MThe Journal of organic chemistry 83(21) 13595-13603 2018年  
  44. Combination Metabolomics Approach for Identifying Endogenous Substrates of Carnitine/Organic Cation Transporter OCTN1.
    Masuo Y, Ohba Y, Yamada K, Al-Shammari AH, Seba N, Nakamichi N, Ogihara T, Kunishima M, Kato YPharmaceutical research 35(11) 224-224 2018年  
  45. Imido-substituted triazines as dehydrative condensing reagents for the chemoselective formation of amides in the presence of free hydroxy groups
    Kitamura Masanori, Sasaki Suguru, Nishikawa Riho, Yamada Kohei, Kunishima MunetakaRSC Advances 8(40) 22482-22489 2018年  
  46. Study of O-Allylation Using Triazine-Based Reagents
    Yamada Kohei, Hayakawa Naoko, Fujita Hikaru, Kitamura Masanori, Kunishima MunetakaChemical & Pharmaceutical Bulletin 65(1) 112-115 2017年  
  47. Phototriggered Dehydration Condensation Using an Aminocyclopropenone
    Mishiro Kenji, Yushima Yuki, Kunishima MunetakaOrganic Letters 19(18) 4912-4915 2017年  
  48. Novel Alkylating Reagents Designed by the Characteristics of 1,3,5-Triazines
    Kunishima Munetaka, Yamada Kohei, Fujita Hikaru, Kitamura MasanoriJournal of Synthetic Organic Chemistry Japan 75(10) 1023-1034 2017年  
  49. N,N ‘-Dimethylated Benzyloxytriazinedione: A Stable Solid Reagent for Acid-Catalyzed O-Benzylation
    Fujita Hikaru, Kakuyama Satoshi, Kunishima MunetakaEuropean Journal of Organic Chemistry (4) 833-839 2017年  
  50. Development of a method for the synthesis of 2,4,5-trisubstituted oxazoles composed of carboxylic acid, amino acid, and boronic acid
    Yamada Kohei, Kamimura Naoto, Kunishima MunetakaBeilstein Journal of Organic Chemistry 13 1478-1485 2017年  
  51. Chemo-enzymatic synthesis of a glycosylated peptide containing a complex N-glycan based on unprotected oligosaccharides by using DMT-MM and Endo-M
    Tomabechi Yusuke, Katoh Toshihiko, Kunishima Munetaka, Inazu Toshiyuki, Yamamoto KenjiGlycoconjugate Journal 34(4) 481-487 2017年  
  52. トリアジンの特性を活用した新規アルキル化剤
    75(10) 1023-1034 2017年  
  53. Potent triazine-based dehydrocondensing reagents substituted by an amido group
    Kunishima Munetaka, Kato Daiki, Kimura Nobu, Kitamura Masanori, Yamada Kohei, Hioki KazuhitoBeilstein Journal of Organic Chemistry 12 1897-1903 2016年  
  54. Mild Amide-Cleavage Reaction Mediated by Electrophilic Benzylation
    Yamada Kohei, Karuo Yukiko, Tsukada Yuichi, Kunishima MunetakaChemistry-a European Journal 22(39) 14042-14047 2016年  
  55. Increased Plasma Concentrations of Unbound SN-38, the Active Metabolite of Irinotecan, in Cancer Patients with Severe Renal Failure
    Fujita Ken-ichi, Masuo Yusuke, Okumura Hidenori, Watanabe Yusuke, Suzuki Hiromichi, Sunakawa Yu, Shimada Ken, Kawara Kaori, Akiyama Yuko, Kitamura Masanori …Pharmaceutical Research 33(2) 269-282 2016年  
  56. Development of acid-catalyzed fluorous benzylating reagents based on a triazinedione core
    Kunishima Munetaka, Asao Ryohei, Yamada Kohei, Kitamura Masanori, Fujita HikaruJournal of Fluorine Chemistry 190 68-74 2016年  
  57. Development of a Triazine-Based tert-Butylating Reagent, TriAT-tBu
    Yamada Kohei, Hayakawa Naoko, Fujita Hikaru, Kitamura Masanori, Kunishima MunetakaEuropean Journal of Organic Chemistry (23) 4093-4098 2016年  
  58. Alcohol- and Amine-Tolerant Synthesis of Six-Membered Cyclic Quaternary Ammonium Salts by Using a Triazine-Based Reagent
    Kitamura Masanori, Yamamura Seina, Yamada Kohei, Kunishima MunetakaAsian Journal of Organic Chemistry 5(12) 1508-1517 2016年  
  59. 125I標識CYP代謝基質誘導体を用いたイメージングによるCYP活性定量法の確立
    水谷明日香, 水谷明日香, 高須啓彰, 外間つづみ, 西井龍一, 鈴木千恵, 小林正和, 北村正典, 国嶋崇隆, 間賀田泰寛 …核医学(Web) 53(Supplement) 1250(J‐STAGE) 2016年  
  60. Study of the Reactivities of Acid-Catalyzed O-Benzylating Reagents Based on Structural Isomers of 1,3,5-Triazine
    Fujita Hikaru, Hayakawa Naoko, Kunishima MunetakaJournal of Organic Chemistry 80(21) 11200-11205 2015年  
  61. O-Benzylation of Carboxylic Acids Using 2,4,6-Tris(benzyloxy)-1,3,5-triazine (TriBOT) under Acidic or Thermal Conditions
    Yamada Kohei, Yoshida Saki, Fujita Hikaru, Kitamura Masanori, Kunishima MunetakaEuropean Journal of Organic Chemistry (36) 7997-8002 2015年  
  62. Synthesis of Pyrrolidinium Salts Using a Triazine-based Reagent under Mild Conditions
    Kitamura Masanori, Yamamura Seina, Kobayashi Hiroko, Yamamoto Mariko, Tada Kayo, Hioki Kazuhito, Yamada Kohei, Kunishima MunetakaChemistry Letters 43(10) 1593-1595 2014年  
  63. Specific Labeling of Streptavidin for Better Understanding of Ligand Modification in Modular Method for Affinity Labeling (MoAL)
    Kunishima Munetaka, Kato Daiki, Nakanishi Shuichi, Kitamura Masanori, Yamada Kohei, Terao Keiji, Asano TomoyaChemical & Pharmaceutical Bulletin 62(11) 1146-1150 2014年  
  64. Role of Linkers in Tertiary Amines That Mediate or Catalyze 1,3,5-Triazine-Based Amide-Forming Reactions
    Kitamura Masanori, Kawasaki Fumitaka, Ogawa Kouichi, Nakanishi Shuichi, Tanaka Hiroyuki, Yamada Kohei, Kunishima MunetakaJournal of Organic Chemistry 79(8) 3709-3714 2014年  
  65. Development of a New Benzylating Reagent Spontaneously Releasing Benzyl Cation Equivalents at Room Temperature
    Yamada Kohei, Tsukada Yuichi, Karuo Yukiko, Kitamura Masanori, Kunishima MunetakaChemistry-a European Journal 20(38) 12274-12278 2014年  
  66. 4-(4,6-Dimethoxy-1,3,5-triazin-2-yl)-4-methylmorpholinium Chloride
    Masanori Kitamura, Munetaka KunishimaEncyclopedia of Reagents for Organic Synthesis 2013年5月  
  67. Synthesis and evaluation of iodinated cyclopropanecarboxylic acid {3-[6-(phenylamino)-pyrimidin-4-ylamino]-phenyl}-amides as EGFR-TK imaging agents
    Yoshimoto Mitsuyoshi, Kimura Sadaaki, Yamada Kohei, Hirata Masahiko, Ohmomo Yoshiro, Kunishima Munetaka, Kawai Keiichi, Fujii HirofumiJournal of Labelled Compounds & Radiopharmaceuticals 56 S373 2013年  
  68. Study of 1,3,5-Triazine-Based Catalytic Amide-Forming Reactions: Effect of Solvents and Basicity of Reactants
    Kunishima Munetaka, Kitamura Masanori, Tanaka Hiroyuki, Nakakura Ichiro, Moriya Takahiro, Hioki KazuhitoChemical & Pharmaceutical Bulletin 61(8) 882-886 2013年  
  69. Binding of sulforhodamine B to human serum albumin: A spectroscopic study
  70. Kitamura Masanori, Murakami Koji, Yamada Kohei, Kawai Keiichi, Kunishima MunetakaDyes and Pigments 99(3) 588-593 2013年  
  71. A Practical Method for p-Methoxybenzylation of Hydroxy Groups Using 2,4,6-Tris(p-methoxybenzyloxy)-1,3,5-triazine (TriBOT-PM)
    Yamada Kohei, Fujita Hikaru, Kitamura Masanori, Kunishima MunetakaSynthesis-Stuttgart 45(21) 2989-2997 2013年  
  72. A new method using 2-chloro-4,6-dimethoxy-1,3,5-triazine for facile elimination of dimethylamino group in Eschenmoser’s methylenation for synthesis of alpha,beta-unsaturated esters
    Yamada Kohei, Masaki Kazumasa, Hagimoto Yuri, Kamiya Seina, Kunishima MunetakaTetrahedron Letters 54(13) 1758-1760 2013年  
  73. Substrate-Selective Dehydrocondensation at the Interface of Micelles and Emulsions of Common Surfactants
    Kunishima Munetaka, Kikuchi Kanako, Kawai Yukio, Hioki KazuhitoAngewandte Chemie-International Edition 51(9) 2080-2083 2012年  
  74. Study on 1,3,5-Triazine Chemistry in Dehydrocondensation: Gauche Effect on the Generation of Active Triazinylammonium Species
    Kunishima Munetaka, Ujigawa Takae, Nagaoka Yoshie, Kawachi Chiho, Hioki Kazuhito, Shiro MotooChemistry-a European Journal 18(49) 15856-15867 2012年  
  75. One-Pot Preparation of Oxazol-5(4H)-ones from Amino Acids in Aqueous Solvents
    Fujita Hikaru, Kunishima MunetakaChemical & Pharmaceutical Bulletin 60(7) 907-912 2012年  
  76. N-Isopropyl-p-iodoamphetamine Hydrochloride Is Predominantly Metabolized by CYP2C19
    Fujita Ken-ichi, Sugiyama Minako, Akiyama Yuko, Hioki Kazuhito, Kunishima Munetaka, Nishi Kodai, Kobayashi Masato, Kawai Keiichi, Sasaki YasutsunaDrug Metabolism and Disposition 40(5) 843-846 2012年  
  77. N-ISOPROPYL-P-IODOAMPHETAMINE HYDROCHLORIDE (IMP) IS PREDOMINANTLY METABOLIZED BY CYP2C19.
    Fujita K, Sugiyama M, Akiyama Y, Hioki K, Kunishima M, Kobayashi M, Kawai K, Sasaki YClinical Pharmacology & Therapeutics 91 S16 2012年  
  78. A Novel Acid-Catalyzed O-Benzylating Reagent with the Smallest Unit of Imidate Structure
    Yamada Kohei, Fujita Hikaru, Kunishima MunetakaOrganic Letters 14(19) 5026-5029 2012年  
  79. New approach to oligotriazoles using a cobalt complex of propargyl azides as a synthetic component
    Tsukada Yuichi, Yamada Kohei, Kunishima MunetakaTetrahedron Letters 52(26) 3358-3360 2011年  
  80. Labeling study of avidin by modular method for affinity labeling (MoAL)
    Nakanishi Shuichi, Tanaka Hiroyuki, Hioki Kazuhito, Yamada Kohei, Kunishima MunetakaBioorganic & Medicinal Chemistry Letters 20(23) 7050-7053 2010年  
  81. Effects of stereochemistry and beta-substituents on the rates of vinylic S(N)2 reaction of hypervalent vinyl(phenyl)-lambda(3)-iodanes with tetrabutylammonium halides
    Miyamoto Kazunori, Okubo Takuji, Hirobe Masaya, Kunishima Munetaka, Ochiai MasahitoTetrahedron 66(31) 5819-5826 2010年  

2010年以前のリストについてはResearchmapを参考にしてください →

北條恵子 講師

  1. Water-Based Solid-Phase Peptide Synthesis without Hydroxy Side Chain Protection
    Keiko Hojo, Yuki Manabe, Tomoyo Uda, Yuko TsudaJOURNAL OF ORGANIC CHEMISTRY 2022年8月  
  2. Environmentally Conscious In-Water Peptide Synthesis Using Boc Strategy
    Keiko Hojo, Suzuko Fujiwara, Hoshito Inai, Yuki Manabe, Yuko TsudaINTERNATIONAL JOURNAL OF PEPTIDE RESEARCH AND THERAPEUTICS 28(2) 2022年3月
  3. Exploration of Active Site-Directed Plasmin Inhibitors: Beyond Tranexamic Acid
    Yuko Tsuda, Koushi Hidaka, Keiko Hojo, Yoshio OkadaPROCESSES 9(2) 2021年2月  
  4. Design of new cyclic plasmin inhibitors
    Yuko Tsuda, Koushi Hidaka, Keiko Hojo, Keigo Gohda, Naoki Teno, Keiko WanakaJOURNAL OF PEPTIDE SCIENCE 24 S117-S118 2018年9月  
  5. Development of a Single-Chain Peptide Agonist of the Relaxin-3 Receptor Using Hydrocarbon Stapling.
    Keiko Hojo, Mohammed Akhter Hossain, Julien Tailhades, Fazel Shabanpoor, Lilian L L Wong, Emma E K Ong-Pålsson, Hanna E Kastman, Sherie Ma, Andrew L Gundlach, K Johan Rosengren …Journal of medicinal chemistry 59(16) 7445-56 2016年8月25日  
  6. Oligomerization of neutral peptides derived from the JC virus agnoprotein through a cysteine residue
    Koushi Hidaka, Keiko Hojo, Shio Fujioka, Souichi Nukuzuma, Yuko TsudaAMINO ACIDS 47(10) 2205-2213 2015年10月  
  7. Development of a Sortase A-mediated Peptide-labeled Liposome Applicable to Drug-delivery Systems.
    Atsushi Tabata, Yukimasa Ohkubo, Natsuki Anyoji, Keiko Hojo, Toshifumi Tomoyasu, Youhei Tatematsu, Kazuto Ohkura, Hideaki NagamuneAnticancer research 35(8) 4411-7 2015年8月  
  8. Aqueous microwave-assisted solid-phase peptide synthesis using Fmoc strategy. III: Racemization studies and water-based synthesis of histidine-containing peptides
    Keiko Hojo, Natsuki Shinozaki, Koushi Hidaka, Yuko Tsuda, Yoshinobu Fukumori, Hideki Ichikawa, John D. WadeAMINO ACIDS 46(10) 2347-2354 2014年10月  
  9. Aqueous Microwave-Assisted Solid-Phase Peptide Synthesis Using Fmoc Strategy. II. Racemization Studies and Water Based Synthesis of Cysteine-Containing Peptides
    Keiko Hojo, Natsuki Shinozaki, Asaki Hara, Mare Onishi, Yoshinobu Fukumori, Hideki IchikawaPROTEIN AND PEPTIDE LETTERS 20(10) 1122-1128 2013年10月  
  10. Aqueous Microwave-Assisted Solid-Phase Synthesis Using Boc-Amino Acid Nanoparticles
    Keiko Hojo, Natsuki Shinozaki, Yoshimi Nozawa, Yoshinobu Fukumori, Hideki IchikawaAPPLIED SCIENCES 3(3) 614-623 2013年9月  
  11. Aqueous microwave-assisted solid-phase peptide synthesis using Fmoc strategy: in-water synthesis of “difficult sequences”.
    Keiko Hojo, Hideki Ichikawa, Asaki Hara, Mare Onishi, Koichi Kawasaki, Yoshinobu FukumoriProtein and peptide letters 19(11) 1231-6 2012年11月  
  12. Development of a method for environmentally friendly chemical peptide synthesis in water using water-dispersible amino acid nanoparticles
    .Keiko Hojo, Asaki Hara, Hiroyuki Kitai, Mare Onishi, Hideki Ichikawa, Yoshinobu Fukumori, Koichi KawasakiChemistry Central journal 5 49-49 2011年8月25日  
  13. Peptide synthesis ‘in water’ by a solution-phase method using water-dispersible nanoparticle Boc-amino acid.
    Keiko Hojo, Hideki Ichikawa, Mare Onishi, Yoshinobu Fukumori, Koichi KawasakiJournal of peptide science : an official publication of the European Peptide Society 17(7) 487-92 2011年7月  
  14. Facile Synthesis of a Chitosan Hybrid of a Laminin-related Peptide and Its Antimetastatic Effect in Mice
    Keiko Hojo, Mitsuko Maeda, Yu Mu, Haruhiko Kamada, Yasuo Tsutsumi, Yasuhiro Nishiy Ama, Tomoko Yoshikawa, Keisuke Kurita, Lawrence H Block, Tadanori Mayumi …Journal of Pharmacy and Pharmacology 52(1) 67-73 2010年2月18日  

2010年以前のリストについてはResearchmapを参考にしてください →